Institut for Lægemiddeldesign og Farmakologi

Kristian Strømgaard

Professor

Biologiske lægemidler
Jagtvej 162
2100 København Ø
- kristian.stromgaard@sund.ku.dk
- https://drug.ku.dk
Telefon: +4535336114

ORCID: 0000-0003-2206-4737

Udgivelsesår:

Alle

76 - 100 ud af 178Pr. side: 25

Sortering: Udgivelsesdato

2015
Udgivet
Identification and characterization of a small-molecule inhibitor of death-associated protein kinase 1
Wilbek, T. S., Skovgaard, T., Sorrell, F. J., Knapp, S., Berthelsen, J. & Strømgaard, Kristian, 2 jan. 2015, I: ChemBioChem. 16, 1, s. 59-63 5 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Binding site residues control inhibitor selectivity in the human norepinephrine transporter but not in the human dopamine transporter
Andersen, J., Ringsted, K. B., Bang-Andersen, B., Strømgaard, Kristian & Kristensen, Anders Skov, 2015, I: Scientific Reports. 5, s. 1-12 12 s., 15650.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Design, Synthesis, and Characterization of Fatty Acid Derivatives of a Dimeric Peptide-Based Postsynaptic Density-95 (PSD-95) Inhibitor
Nissen, K. B., Andersen, J. J., Haugaard-Kedström, L. M., Bach, Anders & Strømgaard, Kristian, 2015, I: Journal of Medicinal Chemistry. 58, s. 1575-1580 6 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Polyamine toxins from spiders and wasps: Polyamine toxins from spiders and wasps
Xiong, X. & Strømgaard, Kristian, 2015, Polyamines: A Universal Molecular Nexus for Growth, Survival, and Specialized Metabolism. Springer, Japan, s. 201-214 14 s.
Publikation: Bidrag til bog/antologi/rapport › Bidrag til bog/antologi › Forskning › fagfællebedømt
Udgivet
Rigidified Clicked Dimeric Ligands for Studying the Dynamics of the PDZ1-2 Supramodule of PSD-95
Eildal, J. N. N., Bach, Anders, Dogan, J., Ye, F., Zhang, M., Jemth, P. & Strømgaard, Kristian, 2015, I: ChemBioChem. 16, s. 64–69 6 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Targeting Protein-Protein Interactions with Trimeric Ligands: High Affinity Inhibitors of the MAGUK Protein Family
Nissen, K. B., Kedström, L. M. H., Wilbek, T. S., Nielsen, L. S., Åberg, E., Kristensen, Anders Skov, Bach, Anders, Jemth, P. & Strømgaard, Kristian, 2015, I: PLOS ONE. 10, 2, s. 1-17 17 s., e0117668.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
2014
Udgivet
Molecular basis of the alternative recruitment of GABA(A) versus glycine receptors through gephyrin
Maric, H., Kasaragod, V. B., Hausrat, T. J., Kneussel, M., Tretter, V., Strømgaard, Kristian & Schindelin, H., 22 dec. 2014, I: Nature Communications. 5, s. 1-11 11 s., 5767.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Structure–Activity Relationship Study of Spider Polyamine Toxins as Inhibitors of Ionotropic Glutamate Receptors
Xiong, X., Poulsen, Mette Homann, Hussein, R. A., Nørager, N. G. & Strømgaard, Kristian, dec. 2014, I: ChemMedChem. 9, 12, s. 2661-70 10 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
THE DEVELOPMENT AND CHARACTERIZATION OF A PEPTIDE-BASED SYNTENIN INHIBITOR - IMPLACATIONS FOR CANCER METASTASIS
Haugaard-Kedstrom, L. M., Albertsen, L., Gil, F. A., Ivarsson, Y., Strømgaard, Kristian & Kedström, L. M. H., sep. 2014, I: Journal of Peptide Science. 20, Suppl. 1, s. s39 1 s., YO11.
Publikation: Bidrag til tidsskrift › Konferenceabstrakt i tidsskrift › Forskning › fagfællebedømt
Udgivet
Mechanistic insight into benzenethiol catalyzed amide bond formations from thioesters and primary amines
Stuhr-Hansen, N., Bork, N. & Strømgaard, Kristian, 14 aug. 2014, I: Organic & Biomolecular Chemistry. 12, 30, s. 5745-51 7 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Structure-activity relationship studies of N-methylated and N-hydroxylated spider polyamine toxins as inhibitors of ionotropic glutamate receptors
Nørager, N. G., Poulsen, Mette Homann, Jensen, A. G., Jeppesen, N. S., Kristensen, Anders Skov & Strømgaard, Kristian, 12 jun. 2014, I: Journal of Medicinal Chemistry. 57, 11, s. 4940-9 10 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Molecular basis for selective serotonin reuptake inhibition by the antidepressant agent fluoxetine (prozac)
Andersen, J., Stuhr-Hansen, N., Zachariassen, L. G., Koldsø, H., Schiøtt, B., Strømgaard, Kristian & Kristensen, Anders Skov, maj 2014, I: Molecular Pharmacology. 85, 5, s. 703-14 12 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Characterization of intracellular regions in the human serotonin transporter for phosphorylation sites
Sørensen, L., Strømgaard, Kristian & Kristensen, Anders Skov, 18 apr. 2014, I: ACS chemical biology. 9, 4, s. 935-44 10 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Inhibition of AMPA Receptors by Polyamine Toxins is Regulated by Agonist Efficacy and Stargazin
Poulsen, Mette Homann, Lucas, S., Strømgaard, Kristian & Kristensen, Anders Skov, 22 feb. 2014, I: Neurochemical Research. 39, 10, s. 1906-1913 8 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Evaluation of PhTX-74 as Subtype-Selective Inhibitor of GluA2-Containing AMPA Receptors
Poulsen, Mette Homann, Lucas, S., Strømgaard, Kristian & Kristensen, Anders Skov, feb. 2014, I: Molecular Pharmacology. 85, 2, s. 261-268 8 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Subunit-Dependent Inhibition of Neuronal Nicotinic Acetylcholine Receptors by Philanthotoxins
Kachel, H. S., Franzyk, Henrik, Strømgaard, Kristian, Tikhonov, D. B. & Mellor, I. R., 28 jan. 2014, I: Biophysical Society. Annual Meeting. Abstracts. 106, 2, s. 338A-338A 1 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning
Udgivet
Facile synthesis of α-hydroxy carboxylic acids from the corresponding α-amino acids
Stuhr-Hansen, N., Padrah, S. & Strømgaard, Kristian, 2014, I: Tetrahedron Letters. 55, 30, s. 4149-4151 3 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Probing backbone hydrogen bonding in PDZ/ligand interactions by protein amide-to-ester mutations
Pedersen, S. W., Pedersen, S. B., Anker, L., Hultqvist, G., Kristensen, Anders Skov, Jemth, P. & Strømgaard, Kristian, 2014, I: Nature Communications. 5, s. 1-11 11 s., 3215.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
The role of backbone hydrogen bonds in the transition state for protein folding of a PDZ domain
Pedersen, S. W., Hultqvist, G., Strømgaard, Kristian & Jemth, P., 2014, I: PLOS ONE. 9, 4, s. 1-7 7 s., e95619.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
2013
Udgivet
Design and synthesis of peptide YY analogues with c-terminal backbone amide-to-ester modifications
Albertsen, L., Andersen, J. J., Paulsson, J. F., Thomsen, J. K., Norrild, J. C. & Strømgaard, Kristian, 12 dec. 2013, I: A C S Medicinal Chemistry Letters. 4, 12, s. 1228-1232 5 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Recombinant production of peptide C-terminal α-amides using an engineered intein
Albertsen, L., Shaw, A. C., Norrild, J. C. & Strømgaard, Kristian, 20 nov. 2013, I: Bioconjugate Chemistry. 24, 11, s. 1883-94 12 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Development of potent fluorescent polyamine toxins and application in labeling of ionotropic glutamate receptors in hippocampal neurons
Nørager, N. G., Jensen, C. B., Rathje, Mette, Andersen, J., Madsen, Kenneth Lindegaard, Kristensen, Anders Skov & Strømgaard, Kristian, 20 sep. 2013, I: A C S Chemical Biology. 8, 9, s. 2033-2041 9 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Probing the role of backbone hydrogen bonds in protein-peptide interactions by amide-to-ester mutations
Eildal, J. N. N., Hultqvist, G., Balle, T., Stuhr-Hansen, N., Padrah, S., Gianni, S., Strømgaard, Kristian & Jemth, P., 4 sep. 2013, I: Journal of the American Chemical Society. 135, 35, s. 12998-3007 10 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
A parallel semisynthetic approach for structure-activity relationship studies of peptide YY
Albertsen, L., Østergaard, S., Paulsson, J. F., Norrild, J. C. & Strømgaard, Kristian, sep. 2013, I: ChemMedChem. 8, 9, s. 1505-13
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Preparation of peptide thioesters through fmoc-based solid-phase peptide synthesis by using amino thioesters
Stuhr-Hansen, N., Wilbek, T. S. & Strømgaard, Kristian, 1 aug. 2013, I: European Journal of Organic Chemistry. 2013, 24, s. 5290-5294 5 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt

Forrige 1 2 3 4 5 6 7 8 Næste

ID: 1302559

Institut for Lægemiddeldesign og Farmakologi

Kristian Strømgaard

Biologiske lægemidler

Identification and characterization of a small-molecule inhibitor of death-associated protein kinase 1

Binding site residues control inhibitor selectivity in the human norepinephrine transporter but not in the human dopamine transporter

Design, Synthesis, and Characterization of Fatty Acid Derivatives of a Dimeric Peptide-Based Postsynaptic Density-95 (PSD-95) Inhibitor

Polyamine toxins from spiders and wasps: Polyamine toxins from spiders and wasps

Rigidified Clicked Dimeric Ligands for Studying the Dynamics of the PDZ1-2 Supramodule of PSD-95

Targeting Protein-Protein Interactions with Trimeric Ligands: High Affinity Inhibitors of the MAGUK Protein Family

Molecular basis of the alternative recruitment of GABA(A) versus glycine receptors through gephyrin

Structure–Activity Relationship Study of Spider Polyamine Toxins as Inhibitors of Ionotropic Glutamate Receptors

THE DEVELOPMENT AND CHARACTERIZATION OF A PEPTIDE-BASED SYNTENIN INHIBITOR - IMPLACATIONS FOR CANCER METASTASIS

Mechanistic insight into benzenethiol catalyzed amide bond formations from thioesters and primary amines

Structure-activity relationship studies of N-methylated and N-hydroxylated spider polyamine toxins as inhibitors of ionotropic glutamate receptors

Molecular basis for selective serotonin reuptake inhibition by the antidepressant agent fluoxetine (prozac)

Characterization of intracellular regions in the human serotonin transporter for phosphorylation sites

Inhibition of AMPA Receptors by Polyamine Toxins is Regulated by Agonist Efficacy and Stargazin

Evaluation of PhTX-74 as Subtype-Selective Inhibitor of GluA2-Containing AMPA Receptors

Subunit-Dependent Inhibition of Neuronal Nicotinic Acetylcholine Receptors by Philanthotoxins

Facile synthesis of α-hydroxy carboxylic acids from the corresponding α-amino acids

Probing backbone hydrogen bonding in PDZ/ligand interactions by protein amide-to-ester mutations

The role of backbone hydrogen bonds in the transition state for protein folding of a PDZ domain

Design and synthesis of peptide YY analogues with c-terminal backbone amide-to-ester modifications

Recombinant production of peptide C-terminal α-amides using an engineered intein

Development of potent fluorescent polyamine toxins and application in labeling of ionotropic glutamate receptors in hippocampal neurons

Probing the role of backbone hydrogen bonds in protein-peptide interactions by amide-to-ester mutations

A parallel semisynthetic approach for structure-activity relationship studies of peptide YY

Preparation of peptide thioesters through fmoc-based solid-phase peptide synthesis by using amino thioesters

Flest downloads

PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions