Institut for Lægemiddeldesign og Farmakologi

Francesco Bavo

Postdoc, Adjunkt

Medicinalkemi
Jagtvej 162, 2100 København Ø
- francesco.bavo@sund.ku.dk
- https://ilf.ku.dk/
Telefon: +4535327264

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Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride
Airoldi, V., Piccolo, O., Roda, G., Appiani, R., Bavo, Francesco, Tassini, R., Paganelli, S., Arnoldi, S., Pallavicini, M. & Bolchi, C., 16 jan. 2020, I: European Journal of Organic Chemistry. 2020, 2, s. 162-168 7 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Structural and stereochemical determinants for hGAT3 inhibition: development of novel conformationally constrained and substituted analogs of (S)-isoserine
Bavo, Francesco, Kickinger, Stefanie, Lie, M. E. K., Avgerinos, Christos, Wilhelmsen, Kristine Sloth, Wellendorph, Petrine & Frølund, Bente, 2023, I: Medicinal Chemistry Research. 32, s. 2299–2324
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype
Bavo, Francesco, Pallavicini, M., Gotti, C., Appiani, R., Moretti, M., Colombo, S. F., Pucci, S., Viani, P., Budriesi, R., Renzi, M., Fucile, S. & Bolchi, C., 24 dec. 2020, I: Journal of Medicinal Chemistry. 63, 24, s. 15668-15692 25 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue
Bavo, Francesco, Pallavicini, M., Pucci, S., Appiani, R., Giraudo, A., Eaton, B., Lucero, L., Gotti, C., Moretti, M., Whiteaker, P. & Bolchi, C., 2022, I: Journal of Medicinal Chemistry. 65, 14, s. 10079-10097
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Determinants for α4β2 vs. α3β4 subtype selectivity of pyrrolidine-based nachrs ligands: A computational perspective with focus on recent cryo-em receptor structures
Bavo, Francesco, Pallavicini, M., Appiani, R. & Bolchi, C., 2021, I: Molecules. 26, 12, 23 s., 3603.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Structure-Activity Studies of 3,9-Diazaspiro[5.5]undecane-Based ?-Aminobutyric Acid Type A Receptor Antagonists with Immunomodulatory Effect
Bavo, Francesco, De-Jong, H., Petersen, Jonas Odgaard, Falk-Petersen, C. B., Löffler, R., Sparrow, E., Rostrup, F., Eliasen, Jannik Nicklas, Wilhelmsen, K. S., Barslund, K., Bundgaard, C., Nielsen, Birgitte, Kristiansen, Uffe, Wellendorph, Petrine, Bogdanov, Y. & Frølund, Bente, 2021, I: Journal of Medicinal Chemistry. 64, 24, s. 17795-17812
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Subnanomolar Affinity and Selective Antagonism at alpha 7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)
Bavo, Francesco, Pallavicini, M., Pucci, S., Appiani, R., Giraudo, A., Oh, H., Kneisley, D. L., Eaton, B., Lucero, L., Gotti, C., Clementi, F., Whiteaker, P. & Bolchi, C., 2023, I: Journal of Medicinal Chemistry. 66, 1, s. 306–332
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry: A review of its recent applications in drug design
Bolchi, C., Bavo, Francesco, Appiani, R., Roda, G. & Pallavicini, M., 15 aug. 2020, I: European Journal of Medicinal Chemistry. 200, 112419.
Publikation: Bidrag til tidsskrift › Review › Forskning › fagfællebedømt
Behavioural and pharmacological profiles of zebrafish administrated pyrrolidinyl benzodioxanes and prolinol aryl ethers with high affinity for heteromeric nicotinic acetylcholine receptors
Braida, D., Ponzoni, L., Moretti, M., Viani, P., Pallavicini, M., Bolchi, C., Appiani, R., Bavo, Francesco, Gotti, C. & Sala, M., 1 aug. 2020, I: Psychopharmacology. 237, 8, s. 2317-2326 10 s.
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Udgivet
Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at gamma-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters
Giraudo, A., Krall, J., Bavo, Francesco, Nielsen, Birgitte, Kongstad, Kenneth Thermann, Rolando, B., De Blasio, R., Gloriam, David E., Löffler, R., Thiesen, L., Harpsøe, Kasper, Frydenvang, Karla Andrea, Boschi, D., Wellendorph, Petrine, Lolli, M. L., Jensen, Anders A. & Frølund, Bente, 27 jun. 2019, I: Journal of Medicinal Chemistry. 62, 12, s. 5797-5809
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt

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ID: 220215448

Institut for Lægemiddeldesign og Farmakologi

Francesco Bavo

Medicinalkemi

Medlem af:

Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride

Structural and stereochemical determinants for hGAT3 inhibition: development of novel conformationally constrained and substituted analogs of (S)-isoserine

Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue

Determinants for α4β2 vs. α3β4 subtype selectivity of pyrrolidine-based nachrs ligands: A computational perspective with focus on recent cryo-em receptor structures

Structure-Activity Studies of 3,9-Diazaspiro[5.5]undecane-Based ?-Aminobutyric Acid Type A Receptor Antagonists with Immunomodulatory Effect

Subnanomolar Affinity and Selective Antagonism at alpha 7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)

1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry: A review of its recent applications in drug design

Behavioural and pharmacological profiles of zebrafish administrated pyrrolidinyl benzodioxanes and prolinol aryl ethers with high affinity for heteromeric nicotinic acetylcholine receptors

Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at gamma-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters

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Exploring the molecular determinants for subtype-selectivity of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogs as betaine/GABA transporter 1 (BGT1) substrate-inhibitors

Subnanomolar Affinity and Selective Antagonism at alpha 7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)